Description

4-Bromo-2-Iodo-7-Azaindole is a high-purity, multi-halogenated heterocyclic building block of significant interest in advanced organic synthesis. Its unique molecular architecture, featuring both bromine and iodine substituents on the 7-azaindole scaffold, makes it a versatile intermediate for constructing complex molecules. This compound is primarily utilized by research chemists and process development scientists in the pharmaceutical and agrochemical industries for applications such as medicinal chemistry, cross-coupling reactions, and the development of novel active ingredients.

Application

• Pharmaceutical Intermediate: Serves as a key precursor in the synthesis of novel drug candidates, particularly in kinase inhibitor research and other targeted therapies.
• Suzuki & Other Cross-Coupling Reactions: The bromine and iodine atoms provide orthogonal reactivity for sequential palladium-catalyzed cross-coupling, enabling the rapid generation of diverse compound libraries.
• Agrochemical Research: Used in the development of new herbicides, fungicides, and insecticides due to the bioactivity of halogenated azaindole derivatives.
• Material Science: Acts as a building block for organic electronic materials, such as organic light-emitting diodes (OLEDs) and semiconductors.
• Chemical Biology & Probe Development: Employed in the creation of molecular probes and tags for studying biological systems and protein interactions.

Basic Information

Product Name	4-Bromo-2-Iodo-7-Azaindole
CAS No.	1260879-70-6
Molecular Formula	C7H4BrIN2
Molecular Weight	322.93 g/mol
Synonyms	4-Bromo-2-iodo-1H-pyrrolo[2,3-b]pyridine; 2-Iodo-4-bromo-7-azaindole; 4-Bromo-2-iodo-1H-7-azaindole; 1H-Pyrrolo[2,3-b]pyridine, 4-bromo-2-iodo-; 4-Br-2-I-7-Azaindole
EINECS	Contact for details

Quality Control

Our 4-Bromo-2-Iodo-7-Azaindole is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing all relevant specifications. Our quality commitment ensures the material meets the high standards required for research and development applications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This compound is light-sensitive (store away from light). Keep away from heat and incompatible materials.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥97.0%
Water Content (KF)	≤0.5%
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.