Description

6-Iodo-3-Nitro-4-Azaindole is a high-purity, advanced pharmaceutical intermediate characterized by its unique halogenated and nitrated azaindole structure. This compound is of significant value for medicinal chemistry research and development, particularly in the synthesis of novel kinase inhibitors and other targeted therapeutic agents. It is primarily utilized by R&D chemists and process development scientists in the pharmaceutical, biotechnology, and fine chemical sectors seeking to build complex heterocyclic scaffolds.

Application

• Pharmaceutical Intermediate: A key building block in the research and synthesis of potential drug candidates, especially kinase inhibitors.
• Medicinal Chemistry Research: Used for structure-activity relationship (SAR) studies and lead optimization in drug discovery programs.
• Chemical Biology Probes: Serves as a precursor for developing molecular probes to study biological pathways and enzyme functions.
• Fine Chemical Synthesis: Employed in multi-step organic synthesis to introduce iodine and nitro functional groups into complex azaindole-based molecules.
• Contract Research & Manufacturing (CRAM): Supplied to organizations offering custom synthesis and process development services.
• Academic Research: Used in university and institutional labs for exploratory research in heterocyclic and organoiodine chemistry.

Basic Information

Product Name	6-Iodo-3-Nitro-4-Azaindole
CAS No.	1260385-30-5
Molecular Formula	C7H4IN3O2
Molecular Weight	289.03 g/mol
Synonyms	4-Azaindole, 6-iodo-3-nitro-; 1H-Pyrrolo[3,2-b]pyridine, 6-iodo-3-nitro-; 3-Nitro-6-iodo-1H-pyrrolo[3,2-b]pyridine; 6-Iodo-3-nitro-1H-pyrrolo[3,2-b]pyridine; 6-Iodo-3-nitropyrrolo[3,2-b]pyridine
EINECS	Contact for details

Quality Control

Every batch of 6-Iodo-3-Nitro-4-Azaindole is produced and tested under a strict quality management system. We ensure compliance with high-purity standards typical for advanced pharmaceutical intermediates. A comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is provided with each shipment to guarantee batch-to-batch consistency and support your regulatory documentation.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at room temperature (15-25°C). Keep the container sealed to protect from moisture.

Specification

Item	Specification
Appearance	Yellow to brown powder or crystalline solid
Identification (HPLC/MS)	Conforms to structure
Purity (HPLC)	≥ 95% (Area %)
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.