Description

(3As,4R,6As)-Rel-2-Boc-Octahydro-Cyclopenta-[C]Pyrrol-4-Carboxylic Acid CAS NO 1251020-10-6 is a high-purity, advanced pharmaceutical intermediate characterized by its complex, stereochemically defined bicyclic structure. This compound is a critical building block in the synthesis of sophisticated active pharmaceutical ingredients (APIs), particularly those targeting the central nervous system. It is essential for research and development chemists and process scale-up teams in the pharmaceutical and biotechnology sectors who require reliable, high-quality intermediates for complex synthetic routes.

Application

• Key Intermediate in API Synthesis: Serves as a crucial chiral scaffold for the production of novel therapeutic agents.
• Neurological & Psychiatric Drug Development: Used in the research and manufacturing of compounds targeting specific neurological receptors and pathways.
• Process Chemistry & Scale-Up: Provides a defined starting point for optimizing and scaling synthetic routes from laboratory to commercial production.
• Medicinal Chemistry Research: Enables the exploration of structure-activity relationships (SAR) in drug discovery programs.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for client-specific projects.
• Production of Stereochemically Complex Molecules: Its defined stereochemistry is leveraged to create molecules with high enantiomeric purity.

Basic Information

Product Name	(3As,4R,6As)-Rel-2-Boc-Octahydro-Cyclopenta-[C]Pyrrol-4-Carboxylic Acid
CAS No.	1251020-10-6
Molecular Formula	C14H23NO4
Molecular Weight	269.34 g/mol
Synonyms	rel-(3aR,4R,6aS)-2-(tert-Butoxycarbonyl)octahydrocyclopenta[c]pyrrole-4-carboxylic Acid; (3aR,4R,6aS)-2-Boc-octahydrocyclopenta[c]pyrrole-4-carboxylic Acid; 2-Boc-4-carboxyhexahydro-1H-cyclopenta[c]pyrrole; tert-Butyl (3aR,4R,6aS)-4-carboxyhexahydro-1H-cyclopenta[c]pyrrole-2(3H)-carboxylate; BOC-Protected Cyclopentapyrrolidine Carboxylic Acid; Advanced Pyrrolidine Intermediate
EINECS	Contact for details

Quality Control

Our production of (3As,4R,6As)-Rel-2-Boc-Octahydro-Cyclopenta-[C]Pyrrol-4-Carboxylic Acid adheres to stringent quality management systems. Every batch undergoes comprehensive analytical testing, including HPLC for purity and chiral analysis, to ensure it meets the exacting standards required for pharmaceutical R&D and manufacturing. Certificates of Analysis (COA) with detailed chromatographic data are provided to guarantee traceability and compliance with your internal specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive); the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Chiral Purity (Chiral HPLC)	≥ 99.0% ee
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Meets ICH Q3C guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.