Description

2-Iodo-6-Methyl-7-Azaindole is a high-purity, halogenated heterocyclic building block of significant interest in advanced organic synthesis. This compound matters as a versatile intermediate for constructing complex molecular architectures, particularly in pharmaceutical research and development. It is primarily needed by medicinal chemists and process development scientists working on kinase inhibitors, targeted cancer therapies, and other bioactive small molecules.

Application

• Pharmaceutical Intermediate: A key synthon for the synthesis of potent kinase inhibitors and other targeted therapeutic agents.
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization campaigns to explore new chemical space.
• Chemical Biology Probes: Serves as a precursor for developing labeled compounds and molecular probes to study biological pathways.
• Agrochemical Research: Potential intermediate in the development of novel active ingredients for crop protection.
• Material Science: Can be utilized in the synthesis of organic electronic materials and functional dyes due to its electron-rich indole core and halogen substituent.

Basic Information

Item	Detail
Product Name	2-Iodo-6-Methyl-7-Azaindole
CAS No.	1227270-88-3
Molecular Formula	C8H7IN2
Molecular Weight	258.06 g/mol
Synonyms	6-Methyl-2-iodo-7-azaindole; 2-Iodo-6-methyl-1H-pyrrolo[2,3-b]pyridine; 1H-Pyrrolo[2,3-b]pyridine, 2-iodo-6-methyl-; 6-Methyl-2-iodo-1H-pyrrolo[2,3-b]pyridine; 2-Iodo-6-methyl-pyrrolo[2,3-b]pyridine
EINECS	Contact for details

Quality Control

Our 2-Iodo-6-Methyl-7-Azaindole is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure high chemical purity and identity confirmation. A comprehensive Certificate of Analysis (COA) detailing purity, impurities, and physical characteristics is provided with every shipment to support your quality assurance protocols.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at room temperature (15-25°C). Keep away from incompatible materials. The product is light-sensitive and should be handled under appropriate conditions to maintain stability.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.