Description

1-(Phenylsulfonyl)-2-Iodo-4-Methoxy-5-Azaindole is a high-purity, functionalized azaindole derivative designed for advanced pharmaceutical and agrochemical research. This compound serves as a critical synthetic intermediate, valued for its unique reactivity profile that enables the construction of complex nitrogen-containing heterocycles. It is primarily utilized by R&D chemists and process development scientists in the life sciences sector for applications in medicinal chemistry, drug discovery, and the synthesis of novel active ingredients.

Application

• Pharmaceutical Intermediate: Key building block in the synthesis of novel drug candidates targeting various therapeutic areas.
• Medicinal Chemistry Research: Used for structure-activity relationship (SAR) studies and lead optimization in drug discovery programs.
• Agrochemical Development: Intermediate in the research and production of new-generation pesticides and herbicides.
• Chemical Biology Probes: Serves as a precursor for developing molecular probes to study biological pathways.
• Material Science Research: Potential monomer or precursor for specialty polymers and advanced organic materials.
• Contract Research & Manufacturing (CRO/CMO): Supplied to service organizations for custom synthesis and scale-up projects.

Basic Information

Product Name	1-(Phenylsulfonyl)-2-Iodo-4-Methoxy-5-Azaindole
CAS No.	1227269-13-7
Molecular Formula	C14H11IN2O3S
Molecular Weight	414.22 g/mol
Synonyms	2-Iodo-4-methoxy-1-(phenylsulfonyl)-1H-pyrrolo[3,2-c]pyridine; 1H-Pyrrolo[3,2-c]pyridine, 2-iodo-4-methoxy-1-(phenylsulfonyl)-; 4-Methoxy-2-iodo-1-(phenylsulfonyl)-1H-pyrrolo[3,2-c]pyridine; 1-(Benzenesulfonyl)-2-iodo-4-methoxy-7-azaindole; 2-Iodo-4-methoxy-1-(phenylsulfonyl)-7-azaindole; 1-(Phenylsulfonyl)-2-iodo-4-methoxy-7-azaindole; 7-Azaindole, 1-(phenylsulfonyl)-2-iodo-4-methoxy- derivative
EINECS	Contact for details

Quality Control

Our 1-(Phenylsulfonyl)-2-Iodo-4-Methoxy-5-Azaindole is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing all critical quality attributes. Our commitment to quality supports compliance with cGMP and ICH guidelines for pharmaceutical intermediates.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated area at a controlled room temperature (15-25°C). Keep away from strong bases and incompatible organic solvents. For long-term storage, consider storage under an inert atmosphere to maintain optimal stability.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.