Description

Mirogabalin CAS NO 1138245-13-2 is a highly selective and potent gabapentinoid compound, functioning as a novel α2δ-1 subunit ligand of voltage-gated calcium channels. Its primary value lies in its targeted mechanism of action, which is critical for the development of next-generation neuropathic pain management therapies. This active pharmaceutical ingredient (API) is essential for pharmaceutical R&D teams and manufacturers focused on creating advanced analgesics for conditions such as diabetic peripheral neuropathy and postherpetic neuralgia.

Application

• Primary Active Pharmaceutical Ingredient (API) for the formulation of prescription medications targeting neuropathic pain.
• Key intermediate in advanced pharmaceutical research and development of novel central nervous system (CNS) therapeutics.
• Reference standard for analytical method development, validation, and quality control in pharmaceutical laboratories.
• Critical material for preclinical and clinical studies investigating new treatments for chronic pain syndromes.
• Used in the synthesis of deuterated or other labeled analogs for metabolic and pharmacokinetic studies.

Basic Information

Product Name	Mirogabalin
CAS No.	1138245-13-2
Molecular Formula	C17H26N2O3
Molecular Weight	306.40 g/mol
Synonyms	Mirogabalin besylate; (1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-ene-6-acetic acid; DS-5565; Tarlige; Gabapentin enacarbil analog; α2δ-1 Ligand; Novel gabapentinoid
EINECS	Contact for details

Quality Control

Our Mirogabalin is manufactured under strict quality management systems to ensure it meets the rigorous standards required for pharmaceutical development. Each batch undergoes comprehensive analytical testing, including identity confirmation, purity assay, and impurity profiling using advanced techniques like HPLC and chiral analysis. A Certificate of Analysis (COA) detailing all specifications and results is provided with every shipment to support your regulatory and R&D documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed in a dry environment to prevent degradation. For long-term storage, consider using desiccants.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to reference standard
Identification (HPLC)	Retention time matches reference
Assay (HPLC)	≥ 98.5%
Chiral Purity	≥ 99.0%
Related Substances (HPLC)	Total impurities ≤ 1.0% Any single impurity ≤ 0.5%
Residual Solvents (GC)	Complies with ICH Q3C
Heavy Metals	≤ 20 ppm
Loss on Drying	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.