Description

4-Cyano-3-Iodo-5-Azaindole is a high-value, multi-functional heterocyclic building block of significant interest in advanced organic synthesis. Its unique molecular architecture, featuring a cyano group, a halogen (iodo) substituent, and an azaindole core, makes it a versatile intermediate for constructing complex pharmacophores. This compound is primarily sought after by research and development teams in the pharmaceutical and agrochemical industries for the discovery and development of novel active ingredients.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of kinase inhibitors and other targeted therapeutic agents, particularly in oncology and antiviral research.
• Agrochemical Research: Used in the development of new herbicides, fungicides, and insecticides, leveraging its heterocyclic scaffold for bioactivity.
• Material Science: Serves as a building block for organic electronic materials and functional dyes due to its electron-deficient aromatic system.
• Chemical Biology: Employed as a molecular probe or a tag in bioconjugation chemistry and proteomics studies.
• Academic & Contract Research: Essential for methodological development in cross-coupling reactions and heterocyclic chemistry within university and CRO laboratories.

Basic Information

Product Name	4-Cyano-3-Iodo-5-Azaindole
CAS No.	1000341-58-1
Molecular Formula	C8H4IN3
Molecular Weight	269.04 g/mol
Synonyms	3-Iodo-1H-pyrrolo[2,3-b]pyridine-4-carbonitrile; 3-Iodo-4-cyano-7-azaindole; 3-Iodo-4-cyano-1H-pyrrolo[2,3-b]pyridine; 4-Cyano-3-iodo-1H-pyrrolo[2,3-b]pyridine; 7-Azaindole-4-carbonitrile, 3-iodo-; 1H-Pyrrolo[2,3-b]pyridine-4-carbonitrile, 3-iodo-
EINECS	Contact for details

Quality Control

Every batch of 4-Cyano-3-Iodo-5-Azaindole is manufactured and tested under a strict quality management system. We provide comprehensive analytical data to ensure the compound meets the high-purity standards required for research and development. A detailed Certificate of Analysis (COA), including results from HPLC, NMR, and mass spectrometry, is supplied with each shipment to guarantee identity, purity, and consistency.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Keep the container sealed to protect from moisture.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.