Description

6-Bromo-3-Iodo-4-Methoxy-5-Azaindole is a high-value, multi-halogenated heterocyclic building block of significant interest in advanced organic synthesis. Its unique structure, featuring bromine and iodine atoms on an azaindole scaffold, makes it a critical intermediate for constructing complex molecular architectures. This compound is primarily utilized by pharmaceutical and agrochemical research organizations for the development of novel active ingredients, including kinase inhibitors and other biologically relevant small molecules.

Application

• Pharmaceutical Intermediate: A key synthon in the research and development of potential drug candidates, particularly for targeted therapies.
• Agrochemical Synthesis: Used in creating novel active ingredients for crop protection products.
• Chemical Biology Probe Development: Serves as a versatile scaffold for designing molecular probes to study biological pathways.
• Material Science Research: Employed in the synthesis of advanced organic electronic materials and ligands for catalysis.
• Cross-Coupling Reactions: The bromo and iodo substituents make it an excellent substrate for Suzuki, Sonogashira, and other palladium-catalyzed cross-coupling reactions.
• Library Synthesis for High-Throughput Screening: Used in combinatorial chemistry to generate diverse compound libraries for biological screening.

Basic Information

Product Name	6-Bromo-3-Iodo-4-Methoxy-5-Azaindole
CAS No.	1000341-19-4
Molecular Formula	C8H6BrIN2O
Molecular Weight	352.96 g/mol
Synonyms	4-Methoxy-6-bromo-3-iodo-1H-pyrrolo[3,2-c]pyridine; 1H-Pyrrolo[3,2-c]pyridine, 6-bromo-3-iodo-4-methoxy-; 6-Bromo-3-iodo-4-methoxy-1H-pyrrolo[3,2-c]pyridine; 5-Azaindole, 6-bromo-3-iodo-4-methoxy-; 4-Methoxy-6-bromo-3-iodo-5-azaindole
EINECS	Contact for details

Quality Control

Our 6-Bromo-3-Iodo-4-Methoxy-5-Azaindole is manufactured under strict quality control protocols to ensure batch-to-batch consistency and high purity for research applications. We provide comprehensive Certificates of Analysis (COA) with each batch, detailing purity, identity, and impurity profiles. Our quality commitment aligns with the standards expected by the pharmaceutical and fine chemical industries.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Keep the container sealed to prevent contamination and moisture absorption.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 95%
Melting Point	Contact for details
Heavy Metals	< 20 ppm
Residual Solvents (GC)	Complies with ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.