Description

5-Chloro-3-Iodo-6-Methyl-7-Azaindole is a high-purity halogenated azaindole derivative, a crucial advanced intermediate in modern pharmaceutical and agrochemical research. Its value lies in its unique molecular scaffold, which serves as a versatile building block for constructing complex molecules with targeted biological activity. This compound is primarily needed by R&D chemists and process development scientists in the pharmaceutical industry for the synthesis of novel drug candidates, particularly in kinase inhibitor and oncology research programs.

Application

• Pharmaceutical Intermediate: A key synthon for the development of kinase inhibitors, anticancer agents, and other small-molecule therapeutics.
• Agrochemical Research: Used in the synthesis of novel herbicides, fungicides, and plant growth regulators.
• Chemical Biology: Serves as a molecular probe or a core structure in fragment-based drug discovery (FBDD).
• Material Science: Potential precursor for organic electronic materials due to its heterocyclic, halogenated structure.
• Custom Synthesis: Employed by contract research and manufacturing organizations (CROs/CMOs) for client-specific projects requiring functionalized azaindoles.
• Academic Research: Utilized in university and institutional labs for methodological studies in heterocyclic and cross-coupling chemistry.

Basic Information

Product Name	5-Chloro-3-Iodo-6-Methyl-7-Azaindole
CAS No.	1000340-16-8
Molecular Formula	C8H6ClIN2
Molecular Weight	292.50 g/mol
Synonyms	5-Chloro-3-iodo-6-methyl-1H-pyrrolo[2,3-b]pyridine; 3-Iodo-5-chloro-6-methyl-7-azaindole; 6-Methyl-5-chloro-3-iodo-7-azaindole; 1H-Pyrrolo[2,3-b]pyridine, 5-chloro-3-iodo-6-methyl-; 5-Chloro-3-iodo-6-methyl-1H-7-azaindole; 5-Chloro-3-iodo-6-methyl-pyrrolo[2,3-b]pyridine
EINECS	Contact for details

Quality Control

Our 5-Chloro-3-Iodo-6-Methyl-7-Azaindole is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing all critical quality attributes. Our production adheres to cGMP principles where applicable, supporting its use in regulated research and development.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, well-ventilated place at a controlled room temperature (15-25°C). Keep the container sealed to minimize exposure to moisture and atmospheric contaminants.

Specification

Item	Specification
Appearance	Off-white to light yellow crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.