Description

Orazipone CAS NO 137109-78-5 is a specialized organic compound belonging to the class of pharmaceutical intermediates. This compound is of significant value in the research and development of novel therapeutic agents, particularly due to its role as a key synthetic building block. It is primarily sought after by pharmaceutical manufacturers and advanced research institutions engaged in drug discovery and process chemistry.

Application

• Pharmaceutical Intermediate: Serves as a critical precursor in the multi-step synthesis of active pharmaceutical ingredients (APIs).
• Drug Discovery Research: Used in medicinal chemistry programs for the design and synthesis of new chemical entities with potential biological activity.
• Process Development & Scale-up: Employed in optimizing synthetic routes for the efficient and cost-effective production of target molecules.
• Reference Standard: Can be utilized as an analytical standard for quality control and method validation in pharmaceutical analysis.
• Biochemical Research: Potential use in studying specific biochemical pathways or as a tool compound in pharmacological assays.

Basic Information

Product Name	Orazipone
CAS No.	137109-78-5
Molecular Formula	C15H12N2O3
Molecular Weight	268.27 g/mol
Synonyms	Orazipone; 5-Methyl-2-phenyl-4H-pyrazolo[1,5-a][1,4]benzodiazepin-4-one; 5-Methyl-2-phenyl-4H-[1,2,4]triazolo[1,5-a][1,4]benzodiazepin-4-one; UNII-8VZR903R6O; 8VZR903R6O; BRN 0970190; CCRIS 6651; LS-132188
EINECS	Contact for details

Quality Control

Our Orazipone is manufactured under a strict quality management system. Every batch undergoes comprehensive analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. A detailed Certificate of Analysis (COA) is provided with each shipment, confirming compliance with agreed specifications. We support cGMP standards for pharmaceutical applications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed to prevent moisture absorption, which may affect stability and handling properties.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (HPLC)	Retention time matches reference standard
Assay (HPLC)	≥ 98.0%
Related Substances (HPLC)	Total impurities ≤ 2.0% Any single impurity ≤ 0.5%
Residual Solvents (GC)	Complies with ICH Q3C guidelines
Loss on Drying	≤ 1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.