Tinib Antineoplastic Drugs

Tinib Antineoplastic Drugs

Tinib antineoplastic drugs are a major class of targeted cancer therapies that inhibit dysregulated tyrosine kinases or serine/threonine kinases involved in tumor growth, angiogenesis, and metastasis. Represented by imatinib, erlotinib, gefitinib, sunitinib, sorafenib, and numerous next-generation inhibitors, these APIs block oncogenic signaling pathways such as EGFR, VEGFR, PDGFR, BCR-ABL, ALK, and RET. Their precision targeting enables high efficacy with reduced systemic toxicity compared to traditional chemotherapy. Tinib drugs are widely used in leukemia, lung cancer, renal cancer, gastrointestinal stromal tumors, and melanoma. Resistance caused by kinase mutations has led to the development of multi-targeted and mutation-specific inhibitors, making tinibs a cornerstone of precision oncology.

Bosutinib Monohydrate CAS NO 918639-08-4

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CAS No.:918639-08-4

Grade:Pharmacy Grade

Content:99.90%

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Bosutinib Methanoate CAS NO 918639-10-8

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CAS No.:918639-10-8

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Content:99.90%

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Ra-9 CAS NO 919091-63-7

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CAS No.:919091-63-7

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Content:99.90%

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2-[(4,7-Dimethyl-2-Quinazolinyl)Amino]-6-(2-Methoxyphenyl)-4(3H)-Pyrimidinone CAS NO 921117-30-8

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CAS No.:921117-30-8

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Content:99.90%

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Refametinib CAS NO 923032-37-5

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CAS No.:923032-37-5

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Content:99.90%

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Nilotinib Hydrochloride Monohydrate CAS NO 923288-90-8

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CAS No.:923288-90-8

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Content:99.90%

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Nilotinib Hydrochloride Anhydrous CAS NO 923288-95-3

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CAS No.:923288-95-3

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Content:99.90%

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Abt-263 CAS NO 923564-51-6

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CAS No.:923564-51-6

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Content:99.90%

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