Description

2-Morpholinopyridine-4-Boronic Acid, Pinacol Ester is a high-value, organoboron building block essential for modern synthetic chemistry, particularly in cross-coupling reactions. Its core value lies in enabling the efficient and selective construction of complex molecules, which is critical for research and development in advanced material and pharmaceutical sciences. This compound is primarily needed by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and material science industries for creating novel active ingredients and functional materials.

Application

• Suzuki-Miyaura Cross-Coupling Reactions: A key reagent for forming carbon-carbon bonds between aromatic rings, fundamental in medicinal chemistry.
• Pharmaceutical Intermediate Synthesis: Used in the research and development of active pharmaceutical ingredients (APIs), especially for kinase inhibitors and other targeted therapies.
• Agrochemical Research: Serves as a building block for creating novel herbicides, fungicides, and insecticides with improved efficacy.
• Material Science & OLED Development: Employed in the synthesis of organic semiconductors, light-emitting materials, and other advanced functional polymers.
• Chemical Biology & Probe Development: Useful for creating molecular probes and labeled compounds for studying biological systems.
• Library Synthesis for Drug Discovery: Facilitates the rapid generation of diverse compound libraries for high-throughput screening.

Basic Information

Product Name	2-Morpholinopyridine-4-Boronic Acid, Pinacol Ester
CAS No.	888721-86-6
Molecular Formula	C15H21BN2O3
Molecular Weight	288.15 g/mol
Synonyms	4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-2-morpholinopyridine; 2-Morpholino-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine; 2-(Morpholin-4-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine; 2-Morpholin-4-ylpyridine-4-boronic acid pinacol ester; 4-Borono-2-morpholinopyridine pinacol ester; 888721-86-6; 2-Morpholinopyridine-4-boronic acid pinacol ester
EINECS	Contact for details

Quality Control

Our 2-Morpholinopyridine-4-Boronic Acid, Pinacol Ester is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity for sensitive synthetic applications. Each lot undergoes rigorous analytical testing, including NMR, HPLC, and mass spectrometry, to confirm identity and purity. Certificates of Analysis (COA) detailing all specifications are available upon request to support your quality assurance and regulatory documentation.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) for long-term storage and when dispensing to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥97.0%
Water Content (KF)	≤0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.