Description

1-(4-Morpholinyl)-2-[4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenoxy]Ethanone is a high-value, multifunctional organic building block that combines a morpholine amide with a protected boronic acid ester. This compound matters as a critical intermediate for modern synthetic chemistry, enabling the precise construction of complex molecules through cross-coupling reactions. It is primarily needed by research and development chemists in the pharmaceutical and agrochemical industries for creating novel active ingredients and advanced materials.

Application

• Pharmaceutical Intermediate: Key building block in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in kinase inhibitor and CNS-active molecule research.
• Agrochemical Synthesis: Used in the development of advanced herbicides, fungicides, and insecticides that require specific aryl-boronate functionalities.
• Material Science Research: Serves as a precursor for organic electronic materials, including polymers and small molecules for OLEDs and OFETs.
• Chemical Biology Probes: Employed in the synthesis of bioconjugates and labeled compounds for proteomics and diagnostic assay development.
• Academic & Contract Research: Essential reagent for methodology development and complex molecule synthesis in academic and CRO laboratories.
• Liquid Crystal & Polymer Chemistry: Intermediate for creating monomers with specific steric and electronic properties for advanced polymeric materials.

Basic Information

Product Name	1-(4-Morpholinyl)-2-[4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenoxy]Ethanone
CAS No.	656257-49-7
Molecular Formula	C18H26BNO5
Molecular Weight	347.22 g/mol
Synonyms	4-(2-Morpholin-4-yl-2-oxoethoxy)phenylboronic acid pinacol ester; 2-Morpholino-2-oxoethyl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl ether; 1-Morpholino-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy]ethan-1-one; 4-[2-Oxo-2-(morpholin-4-yl)ethoxy]benzeneboronic acid pinacol ester; 656257-49-7; 2-(4-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)phenoxy)-1-morpholinoethanone
EINECS	Contact for details

Quality Control

Our 1-(4-Morpholinyl)-2-[4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenoxy]Ethanone is manufactured under strict quality management systems. Every batch undergoes rigorous analytical testing, including HPLC, NMR, and MS, to ensure high purity and structural identity. Certificates of Analysis (COA) with full analytical data are provided to guarantee compliance with your research and production specifications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent moisture absorption and decomposition.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.