Description

5-Bromo-2,6-Dimethoxypyridine-3-Boronic Acid is a high-purity boronic acid derivative and a valuable synthetic building block. Its core value lies in its dual functionality, serving as a key intermediate in the synthesis of complex molecules via cross-coupling reactions. This compound is primarily needed by R&D chemists and process development scientists in the pharmaceutical and agrochemical industries for constructing novel active ingredients.

Application

• Pharmaceutical Intermediate: A crucial building block in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in kinase inhibitor and antiviral research.
• Agrochemical Synthesis: Used to create advanced pyridine-based herbicides, fungicides, and insecticides with improved efficacy and selectivity.
• Material Science Research: Employed in the development of organic electronic materials, such as ligands for metal-organic frameworks (MOFs) or components for organic semiconductors.
• Chemical Biology Probes: Serves as a precursor for synthesizing tagged molecules or inhibitors used to study biological pathways and protein functions.
• Custom Synthesis & Contract Manufacturing: A key starting material for custom synthesis houses and CDMOs (Contract Development and Manufacturing Organizations) producing bespoke compounds for clients.
• Academic Research: Utilized in university and institutional labs for methodological development in organic synthesis and catalysis studies.

Basic Information

Item	Details
Product Name	5-Bromo-2,6-Dimethoxypyridine-3-Boronic Acid
CAS No.	2121513-61-7
Molecular Formula	C7H9BBrNO4
Molecular Weight	261.87 g/mol
Synonyms	(5-Bromo-2,6-dimethoxypyridin-3-yl)boronic acid; 3-Borono-5-bromo-2,6-dimethoxypyridine; 5-Bromo-2,6-dimethoxy-3-pyridineboronic acid; 5-Bromo-2,6-dimethoxypyridine-3-boronic acid pinacol ester (protected form); 2121513-61-7; 5-Br-2,6-(OMe)2-Py-3-B(OH)2
EINECS	Contact for details

Quality Control

Our 5-Bromo-2,6-Dimethoxypyridine-3-Boronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and NMR for structural confirmation, to ensure it meets the high standards required for advanced synthetic applications. A comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). This compound is moisture-sensitive (hygroscopic); keep the container tightly sealed under an inert atmosphere (e.g., nitrogen or argon) for long-term storage to maintain optimal purity and reactivity.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Heavy Metals	≤ 20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.