Description

2-(Morpholin-4-Ylmethyl)Benzeneboronic Acid is a specialized organoboron compound featuring a benzeneboronic acid core functionalized with a morpholinomethyl substituent. This structure makes it a valuable key synthetic intermediate in modern organic and medicinal chemistry, particularly in cross-coupling reactions. It is primarily used by researchers and manufacturers in the pharmaceutical and agrochemical industries for the development of novel active ingredients and complex molecules.

Application

• Pharmaceutical Intermediate: A crucial building block in Suzuki-Miyaura cross-coupling reactions for synthesizing biaryl structures found in drug candidates.
• Agrochemical Synthesis: Used in the research and production of advanced pesticides and herbicides requiring specific aryl-aryl linkages.
• Material Science Research: Serves as a monomer or functionalization agent in the development of organic electronic materials and polymers.
• Chemical Biology & Proteomics: Employed as a probe or linker molecule due to the boronic acid group's affinity for diols.
• Catalyst Ligand Precursor: Can be utilized to develop novel ligand systems for transition metal catalysis.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs for the production of bespoke, high-value chemical entities.

Basic Information

Product Name	2-(Morpholin-4-Ylmethyl)Benzeneboronic Acid
CAS No.	223433-45-2
Molecular Formula	C₁₁H₁₆BNO₃
Molecular Weight	221.06 g/mol
Synonyms	2-(Morpholinomethyl)phenylboronic Acid; [2-(Morpholin-4-ylmethyl)phenyl]boronic Acid; 2-(4-Morpholinylmethyl)benzeneboronic Acid; B-[2-(4-Morpholinylmethyl)phenyl]boronic Acid; 2-Morpholin-4-ylmethyl-benzeneboronic Acid; (2-((Morpholin-4-yl)methyl)phenyl)boronic Acid; 223433-45-2; 2-(Morpholinomethyl)benzeneboronic acid pinacol ester (related ester)
EINECS	Contact for details

Quality Control

Every batch of 2-(Morpholin-4-Ylmethyl)Benzeneboronic Acid is produced and tested under a strict quality management system. We provide comprehensive analytical data to ensure the material meets the high-purity standards required for sensitive synthetic applications. A Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is supplied with each shipment to guarantee traceability and consistency for your R&D and production needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This material is hygroscopic (moisture-sensitive) and should be handled under a dry inert atmosphere to maintain stability and purity. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder or crystalline solid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥95% (Typical 97-99%)
Water Content (KF)	≤1.0%
Heavy Metals	<20 ppm

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.