Description

(2-(4-Methylpiperidin-1-Yl)Pyrimidin-5-Yl)Boronic Acid is a high-purity boronic acid derivative, a crucial building block in modern synthetic chemistry. Its core value lies in enabling the efficient construction of complex molecules through reliable cross-coupling reactions. This advanced intermediate is primarily needed by research and development teams in the pharmaceutical and agrochemical industries for drug discovery and the synthesis of novel active ingredients.

Application

• Pharmaceutical Intermediate: A key precursor in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in kinase inhibitor and other small-molecule therapeutic programs.
• Agrochemical Research: Used in the development of new pesticides and herbicides, where the pyrimidine and piperidine motifs are common pharmacophores.
• Material Science: Serves as a functional monomer or linker in the synthesis of advanced organic materials, such as metal-organic frameworks (MOFs) or polymers with specific electronic properties.
• Chemical Biology & Probe Development: Employed in the creation of molecular probes and bioconjugates for studying biological pathways and target engagement.
• Catalyst Ligand Synthesis: Acts as a starting material for the preparation of sophisticated ligands used in homogeneous catalysis.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for the production of bespoke compounds at various scales.

Basic Information

Product Name	(2-(4-Methylpiperidin-1-Yl)Pyrimidin-5-Yl)Boronic Acid
CAS No.	1704073-33-5
Molecular Formula	C10H16BN3O2
Molecular Weight	221.07 g/mol
Synonyms	5-Pyrimidineboronic acid, 2-(4-methyl-1-piperidinyl)-; 2-(4-Methylpiperidin-1-yl)pyrimidine-5-boronic acid; (2-(4-Methyl-1-piperidinyl)-5-pyrimidinyl)boronic acid; B-[2-(4-Methyl-1-piperidinyl)-5-pyrimidinyl]boronic acid; 1704073-33-5; Boronic acid, B-[2-(4-methyl-1-piperidinyl)-5-pyrimidinyl]-; AKOS025146064; FT-0697605
EINECS	Contact for details

Quality Control

Our (2-(4-Methylpiperidin-1-Yl)Pyrimidin-5-Yl)Boronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. Certificates of Analysis (COA) documenting all specifications are provided and available upon request, supporting compliance in regulated research and development environments.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥95% (Anhydrous basis)
Water Content (KF)	≤1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.