Description

4-Methyl-2-(Piperidin-4-Ylmethoxy)-5-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Pyridine is a high-value, multi-functional boronic ester derivative designed for advanced organic synthesis and pharmaceutical research. This compound is a critical building block for constructing complex molecules via cross-coupling reactions, offering significant advantages in drug discovery pipelines. It is primarily sought by pharmaceutical R&D teams and fine chemical manufacturers developing novel therapeutic agents.

Application

• Suzuki-Miyaura Cross-Coupling Reactions: A key reagent for forming carbon-carbon bonds in the synthesis of complex biaryl and heterobiaryl structures.
• Pharmaceutical Intermediate: Serves as a crucial precursor in the research and development of new active pharmaceutical ingredients (APIs), particularly in oncology and CNS drug candidates.
• Medicinal Chemistry: Used extensively in lead optimization and structure-activity relationship (SAR) studies to explore novel chemical space.
• Chemical Biology Probes: Enables the synthesis of tagged molecules for studying biological pathways and target engagement.
• Agrochemical Research: Employed in the development of new herbicides and fungicides that require specific boronic ester functionalities.
• Material Science: Potential building block for creating organic electronic materials and metal-organic frameworks (MOFs).

Basic Information

Item	Detail
Product Name	4-Methyl-2-(Piperidin-4-Ylmethoxy)-5-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Pyridine
CAS No.	1350559-11-3
Molecular Formula	C19H29BN2O3
Molecular Weight	344.26 g/mol
Synonyms	4-Methyl-2-((piperidin-4-yl)methoxy)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine; 2-(Piperidin-4-ylmethoxy)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4-methylpyridine; 1350559-11-3; 4-Methyl-2-(piperidin-4-ylmethoxy)-5-(tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine; Pinacol ester of (6-Methyl-3-((piperidin-4-yl)methoxy)pyridin-2-yl)boronic acid
EINECS	Contact for details

Quality Control

Our 4-Methyl-2-(Piperidin-4-Ylmethoxy)-5-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Pyridine is manufactured under strict quality systems to ensure batch-to-batch consistency and high purity suitable for research and development. All products undergo rigorous analytical testing, including HPLC, NMR, and MS, to confirm identity and purity. A comprehensive Certificate of Analysis (COA) detailing all specifications is provided with each shipment to support your quality assurance protocols.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent moisture absorption and degradation.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 95%
Water Content (KF)	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.