Description

5-Methoxy-1-Methyl-2-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)-1H-Indole is a high-value, synthetically versatile indole-based boronic ester building block, essential for modern cross-coupling reactions. Its core value lies in enabling the efficient and selective construction of complex molecular architectures, which is critical for research and development in advanced chemistry. This compound is primarily needed by pharmaceutical R&D teams, agrochemical innovators, and specialty chemical manufacturers focused on creating novel active ingredients and functional materials.

Application

• Pharmaceutical Intermediate: A key precursor in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in oncology and CNS therapeutic areas.
• Agrochemical Synthesis: Used to construct complex heterocyclic scaffolds found in next-generation herbicides, fungicides, and insecticides.
• Material Science Research: Serves as a building block for creating organic electronic materials, such as OLED emitters and charge-transport layers.
• Chemical Biology & Probe Development: Employed in the synthesis of fluorescent tags and molecular probes for studying biological systems.
• Academic & Contract Research: A valuable reagent for methodological development in organic synthesis and catalysis studies at universities and CROs.
• Fine Chemical Production: Integral to the multi-step synthesis of complex fragrance and flavor ingredients.

Basic Information

Item	Details
Product Name	5-Methoxy-1-Methyl-2-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)-1H-Indole
CAS No.	1256360-41-4
Molecular Formula	C16H22BNO3
Molecular Weight	287.16 g/mol
Synonyms	2-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-5-methoxy-1-methyl-1H-indole; 5-Methoxy-1-methyl-1H-indole-2-boronic acid pinacol ester; 1-Methyl-5-methoxyindole-2-boronic acid pinacol ester; 5-Methoxy-1-methylindole-2-boronic acid pinacol ester; 1H-Indole-2-boronic acid, 5-methoxy-1-methyl-, 4,4,5,5-tetramethyl-1,3,2-dioxaborolane ester; 5-MeO-1-Me-2-Bpin-indole
EINECS	Contact for details

Quality Control

Our 5-Methoxy-1-Methyl-2-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)-1H-Indole is manufactured under strict quality management systems. Every batch undergoes rigorous analytical testing, including HPLC, NMR, and GC-MS, to ensure high purity and consistency. Certificates of Analysis (COA) detailing identity, purity, and impurity profiles are provided with each shipment to support your quality assurance and regulatory needs.

Storage

Preserve in a tightly closed container, protected from light. Store under an inert atmosphere (e.g., nitrogen or argon) at a controlled room temperature (15-25°C) in a cool, dry, and well-ventilated place. Keep away from oxidizing agents and strong acids.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.