Description

4-(1-Piperidinylmethyl)Phenylboronic Acid is a specialized organoboron compound featuring a phenylboronic acid core functionalized with a piperidinylmethyl group. This structural motif makes it a valuable building block in modern synthetic organic chemistry, particularly for cross-coupling reactions. It is primarily utilized by pharmaceutical and agrochemical research organizations for the development of novel active ingredients and complex molecular architectures.

Application

• Suzuki-Miyaura Cross-Coupling Reactions: A key reagent for forming carbon-carbon bonds in the synthesis of biaryl compounds, a common scaffold in drug discovery.
• Pharmaceutical Intermediate: Serves as a critical precursor in the research and development of new therapeutic agents, including kinase inhibitors and CNS-active compounds.
• Agrochemical Synthesis: Used in creating advanced active ingredients for crop protection products.
• Material Science Research: Employed in the synthesis of organic electronic materials and functional polymers.
• Chemical Biology Probes: Utilized in the development of molecular probes and sensors due to its boronic acid functionality.
• Catalyst Ligand Preparation: Acts as a precursor for synthesizing novel ligands used in homogeneous catalysis.

Basic Information

Product Name	4-(1-Piperidinylmethyl)Phenylboronic Acid
CAS No.	1200434-84-9
Molecular Formula	C13H20BNO2
Molecular Weight	233.12 g/mol
Synonyms	[4-(Piperidin-1-ylmethyl)phenyl]boronic acid; 4-(Piperidin-1-ylmethyl)benzeneboronic acid; 1-[4-(Boronophenyl)methyl]piperidine; 4-(Piperidinomethyl)phenylboronic acid; 4-(1-Piperidinylmethyl)benzeneboronic Acid; 4-Piperidin-1-ylmethyl-phenylboronic acid; B-[4-(1-Piperidinylmethyl)phenyl]boronic acid
EINECS	Contact for details

Quality Control

Our 4-(1-Piperidinylmethyl)Phenylboronic Acid is produced under strict quality management protocols. Each batch undergoes rigorous analytical testing, including HPLC for purity and NMR for structural confirmation, to ensure it meets the high standards required for research and development applications. A comprehensive Certificate of Analysis (COA) detailing identity, purity, and impurity profiles is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and must be kept under an inert atmosphere (e.g., nitrogen or argon) for long-term storage to maintain stability and purity.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 1.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.