Description

2-(n-Methylaminomethyl)Phenylboronic Acid,Pinacol Ester is a specialized organoboron compound featuring a protected boronic acid group and a methylaminomethyl side chain. This unique structure makes it a valuable advanced pharmaceutical intermediate and a versatile building block in modern synthetic chemistry. It is primarily utilized by researchers and manufacturers in the pharmaceutical, agrochemical, and material science industries for the development of novel active ingredients and functional molecules.

Application

• Suzuki-Miyaura Cross-Coupling Reactions: A key reagent for forming carbon-carbon bonds in the synthesis of complex biaryl structures, crucial for drug discovery.
• Pharmaceutical Intermediate: Serves as a critical building block in the synthesis of active pharmaceutical ingredients (APIs), particularly for targeted therapies.
• Agrochemical Synthesis: Used in the research and development of new herbicides, fungicides, and insecticides with improved efficacy.
• Material Science Research: Employed in the creation of organic electronic materials, sensors, and metal-organic frameworks (MOFs).
• Chemical Biology & Proteomics: Acts as a functional handle for bioconjugation and the development of chemical probes.
• Catalyst Ligand Precursor: Can be modified to create novel ligands for transition metal catalysis.

Basic Information

Product Name	2-(n-Methylaminomethyl)Phenylboronic Acid,Pinacol Ester
CAS No.	1150271-47-8
Molecular Formula	C15H24BNO2
Molecular Weight	261.17 g/mol
Synonyms	2-[(Methylamino)methyl]benzeneboronic acid pinacol ester; (2-((Methylamino)methyl)phenyl)boronic acid pinacol ester; N-Methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzylamine; 2-(Methylaminomethyl)phenylboronic acid pinacol ester; B-[2-[(Methylamino)methyl]phenyl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane; CAS 1150271-47-8
EINECS	Contact for details

Quality Control

Our production of 2-(n-Methylaminomethyl)Phenylboronic Acid,Pinacol Ester adheres to stringent quality management protocols. Every batch undergoes comprehensive analytical testing, including HPLC, NMR, and GC, to ensure identity, purity, and consistency. A detailed Certificate of Analysis (COA) is provided with each shipment, confirming compliance with agreed specifications. We support cGMP and ISO standards for pharmaceutical and industrial applications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) for long-term storage or when opening the container to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.