Description

(4-Methoxy-3-(Morpholinosulfonyl)Phenyl)Boronic Acid is a high-purity boronic acid derivative featuring a morpholinosulfonyl substituent, a key structural motif for advanced chemical synthesis. This compound matters as a sophisticated building block in cross-coupling reactions, enabling the precise construction of complex molecules for research and development. It is primarily needed by pharmaceutical and agrochemical R&D teams, as well as academic researchers, for creating novel active ingredients and functional materials.

Application

• Pharmaceutical Intermediate: A crucial building block in Suzuki-Miyaura cross-coupling reactions for synthesizing novel drug candidates, particularly in kinase inhibitor and other small-molecule therapeutic programs.
• Agrochemical Research: Used in the development of new herbicides, fungicides, and insecticides by enabling the introduction of the (4-Methoxy-3-(Morpholinosulfonyl)Phenyl) moiety into target structures.
• Material Science: Serves as a monomer or functionalization agent in the synthesis of advanced polymers, organic electronic materials, and metal-organic frameworks (MOFs).
• Chemical Biology & Proteomics: Acts as a probe or linker in bioconjugation chemistry due to the specific reactivity of the boronic acid group with diols and other functional groups.
• Catalyst & Ligand Development: Utilized as a precursor for creating novel palladium catalysts or bidentate ligands for asymmetric synthesis.
• Academic & Contract Research: Employed in university and CRO laboratories for methodological development in organic synthesis and medicinal chemistry projects.

Basic Information

Product Name	(4-Methoxy-3-(Morpholinosulfonyl)Phenyl)Boronic Acid
CAS No.	1100095-14-4
Molecular Formula	C11H16BNO6S
Molecular Weight	301.13 g/mol
Synonyms	4-Methoxy-3-(morpholine-4-sulfonyl)benzeneboronic acid; 3-(Morpholinosulfonyl)-4-methoxybenzeneboronic acid; [4-Methoxy-3-(morpholine-4-sulfonyl)phenyl]boronic acid; B-[4-Methoxy-3-(4-morpholinesulfonyl)phenyl]boronic acid; (4-Methoxy-3-morpholinosulfonylphenyl)boronic Acid; 1100095-14-4; AKOS025247065
EINECS	Contact for details

Quality Control

Our (4-Methoxy-3-(Morpholinosulfonyl)Phenyl)Boronic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. Certificates of Analysis (COA) detailing all specifications are provided with every shipment. We support cGMP and ISO standards for pharmaceutical and industrial applications.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under an inert atmosphere (e.g., nitrogen or argon) for long-term storage to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥97.0% (Area %)
Water Content (KF)	≤1.0%
Heavy Metals	≤20 ppm
Residue on Ignition	≤0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.