Description

1-(4-Morpholinyl)-2-[4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenyl]-Ethanone is a high-value boronic ester derivative, serving as a critical synthetic intermediate in modern organic chemistry. Its core value lies in enabling efficient Suzuki-Miyaura cross-coupling reactions, a cornerstone methodology for constructing complex biaryl and heterobiaryl structures. This compound is essential for researchers and manufacturers in the pharmaceutical, agrochemical, and advanced materials sectors who require reliable, high-purity building blocks for drug discovery and specialty chemical synthesis.

Application

• Pharmaceutical Intermediate: Key building block for the synthesis of active pharmaceutical ingredients (APIs) and drug candidates, particularly those containing morpholine and biaryl motifs.
• Agrochemical Synthesis: Used in the research and development of novel herbicides, fungicides, and insecticides that require specific aryl-aryl linkages.
• Material Science Research: Serves as a precursor for organic electronic materials, including ligands for OLEDs and components for organic semiconductors.
• Chemical Biology & Proteomics: Employed in the synthesis of molecular probes and bioconjugation reagents for studying biological systems.
• Academic & Industrial R&D: A versatile reagent for method development and library synthesis in medicinal and process chemistry laboratories.
• Custom Synthesis & Contract Manufacturing: Supplied as a high-purity starting material for custom chemical synthesis and scale-up projects.

Basic Information

Item	Details
Product Name	1-(4-Morpholinyl)-2-[4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenyl]-Ethanone
CAS No.	1092563-23-9
Molecular Formula	C18H26BNO4
Molecular Weight	331.22 g/mol
Synonyms	4'-(Morpholin-4-ylacetyl)phenylboronic acid pinacol ester; 2-[4-(4-Morpholinylacetyl)phenyl]-4,4,5,5-tetramethyl-1,3,2-dioxaborolane; 1-Morpholino-2-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]ethanone; 4-(2-Morpholino-2-oxoethyl)phenylboronic acid pinacol ester; (4-(2-Morpholino-2-oxoethyl)phenyl)boronic acid pinacol ester
EINECS	Contact for details

Quality Control

Our 1-(4-Morpholinyl)-2-[4-(4,4,5,5-Tetramethyl-1,3,2-Dioxaborolan-2-Yl)Phenyl]-Ethanone is produced under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and LC-MS, to ensure high chemical purity and structural identity. Certificates of Analysis (COA) with detailed specifications are provided and available upon request to support your quality assurance and regulatory documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.