Description

6-(Morpholin-4-Ylamino)Pyridine-3-Boronic Acid Pinacol Ester is a high-purity, organoboron building block designed for advanced pharmaceutical and agrochemical research. This compound matters because it serves as a critical intermediate in Suzuki-Miyaura cross-coupling reactions, enabling the efficient synthesis of complex molecules. It is primarily needed by medicinal chemists and process development scientists in the pharmaceutical, agrochemical, and material science industries for constructing novel chemical entities.

Application

• Pharmaceutical Intermediate: Key building block for the synthesis of active pharmaceutical ingredients (APIs) and drug candidates via palladium-catalyzed cross-coupling.
• Agrochemical Research: Used in the development of novel herbicides, fungicides, and insecticides requiring specific heterocyclic architectures.
• Material Science: Employed in the creation of organic electronic materials, such as polymers and small molecules for OLEDs and OFETs.
• Chemical Biology: Serves as a probe or linker in the development of biochemical tools and PROTACs (Proteolysis Targeting Chimeras).
• Catalyst Ligand Synthesis: A precursor for synthesizing novel ligand systems used in homogeneous catalysis.
• Custom Synthesis & Contract Manufacturing: Supplied to CDMOs (Contract Development and Manufacturing Organizations) for custom synthesis projects.

Basic Information

Product Name	6-(Morpholin-4-Ylamino)Pyridine-3-Boronic Acid Pinacol Ester
CAS No.	1073354-38-7
Molecular Formula	C15H24BN3O3
Molecular Weight	305.18 g/mol
Synonyms	6-(4-Morpholinylamino)-3-pyridineboronic acid pinacol ester; 6-Morpholin-4-ylaminopyridine-3-boronic acid pinacol ester; 6-(N-Morpholino)aminopyridine-3-boronic acid pinacol ester; 3-Pyridineboronic acid, 6-[(4-morpholinyl)amino]-, 1,1-dimethylethyl ester; (6-(Morpholin-4-ylamino)pyridin-3-yl)boronic acid pinacol ester; PINACOL 6-(MORPHOLINOAMINO)PYRIDIN-3-YLBORONATE
EINECS	Contact for details

Quality Control

Our 6-(Morpholin-4-Ylamino)Pyridine-3-Boronic Acid Pinacol Ester is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure high purity and batch-to-batch consistency suitable for sensitive coupling reactions. A comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is moisture-sensitive (hygroscopic); keep the container tightly sealed under an inert atmosphere (argon or nitrogen) for long-term storage to maintain stability and purity.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (HPLC)	Conforms
Identification (NMR)	Conforms
Purity (HPLC)	≥97.0%
Water Content (KF)	≤0.5%
Residue on Ignition	≤0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.