Description

[2-([1,3,2]Dioxaborinan-2-Yloxy)-Ethyl]-Dimethyl-Amine is a specialized organoboron compound featuring a dioxaborinane ring linked to a tertiary amine via an ethoxy spacer. This unique structure makes it a valuable bifunctional reagent, serving as both a protected boronic acid equivalent and a source of a dimethylaminoethyl group for chemical synthesis. It is primarily utilized as a key intermediate and building block in advanced pharmaceutical research, agrochemical development, and materials science.

Application

• Pharmaceutical Intermediate: A crucial building block in the synthesis of active pharmaceutical ingredients (APIs), particularly for boron-containing drugs and protease inhibitors.
• Suzuki-Miyaura Cross-Coupling: Acts as a stable, protected boronic ester reagent for palladium-catalyzed cross-coupling reactions to form carbon-carbon bonds.
• Agrochemical Synthesis: Used in the research and production of novel herbicides, fungicides, and insecticides that incorporate boron or amine functionalities.
• Polymer & Material Science: Serves as a monomer or functionalization agent for creating specialty polymers, coatings, and boron nitride precursors.
• Ligand & Catalyst Development: Employed in the design and synthesis of novel chelating ligands and organocatalysts.
• Bioconjugation & Labeling: Useful for modifying biomolecules, peptides, or surfaces due to its reactive amine and protected boronate groups.

Basic Information

Product Name	[2-([1,3,2]Dioxaborinan-2-Yloxy)-Ethyl]-Dimethyl-Amine
CAS No.	13368-62-2
Molecular Formula	C7H16BNO3
Molecular Weight	173.02 g/mol
Synonyms	2-(2-(Dimethylamino)ethoxy)-1,3,2-dioxaborinane; N,N-Dimethyl-2-(1,3,2-dioxaborinan-2-yloxy)ethanamine; (2-(Dimethylamino)ethoxy)boronic acid, cyclic ester; 2-(2-Dimethylaminoethoxy)-1,3,2-dioxaborinane; Dimethyl-[2-(1,3,2-dioxaborinan-2-yloxy)-ethyl]-amine; 2-(N,N-Dimethylaminoethyloxy)-1,3,2-dioxaborinane
EINECS	Contact for details

Quality Control

Our [2-([1,3,2]Dioxaborinan-2-Yloxy)-Ethyl]-Dimethyl-Amine is produced under strict quality management systems. Every batch undergoes rigorous analytical testing to ensure high purity and consistency, meeting the stringent requirements for research and industrial synthesis. Comprehensive Certificates of Analysis (COA) detailing purity, identity, and impurity profiles are provided with each shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed under an inert atmosphere (e.g., nitrogen or argon) after opening to prevent degradation.

Specification

Item	Specification
Appearance	Colorless to pale yellow liquid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.