Description

5-(4-Morpholinylmethyl)-3-Furoic Acid is a specialized heterocyclic building block of significant interest in advanced organic synthesis. This compound matters for its unique molecular architecture, which combines a furan carboxylic acid moiety with a morpholine substituent, enabling precise modifications in complex molecule construction. Pharmaceutical research and development teams, particularly those focused on medicinal chemistry and the creation of novel active pharmaceutical ingredients (APIs), are the primary industrial users of this high-value intermediate.

Application

• Pharmaceutical Intermediate: Serves as a key synthon in the research and development of new drug candidates, particularly for central nervous system (CNS) and anti-infective targets.
• Medicinal Chemistry: Used as a versatile scaffold for structure-activity relationship (SAR) studies and lead optimization due to its modifiable acid and amine functional groups.
• Organic Synthesis Building Block: Employed in the construction of complex heterocyclic compounds, including fused ring systems and functionalized molecules for material science.
• Agrochemical Research: Potential application in the synthesis of novel crop protection agents and herbicides.
• Ligand and Catalyst Development: The morpholine and carboxylic acid groups make it a candidate for developing chelating ligands or organocatalysts.

Basic Information

Product Name	5-(4-Morpholinylmethyl)-3-Furoic Acid
CAS No.	932854-92-7
Molecular Formula	C10H13NO4
Molecular Weight	211.21 g/mol
Synonyms	3-Furoic acid, 5-[(4-morpholinyl)methyl]-; 5-(Morpholin-4-ylmethyl)furan-3-carboxylic acid; 5-(4-Morpholinylmethyl)-3-furancarboxylic acid; 932854-92-7; 5-(Morpholinomethyl)-3-furoic acid; 4-[(3-Carboxyfuran-5-yl)methyl]morpholine
EINECS	Contact for details

Quality Control

Our 5-(4-Morpholinylmethyl)-3-Furoic Acid is produced under strict quality management systems to ensure batch-to-batch consistency and high purity, suitable for demanding research applications. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing key parameters such as assay, identity, and impurity profiles. Our quality commitment aligns with cGMP principles for pharmaceutical intermediates, ensuring traceability and reliability for our global partners.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Keep away from strong acids and incompatible materials such as strong oxidizing agents. For long-term storage, consider storing under an inert atmosphere to maintain optimal stability.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Related Substances (HPLC)	Total impurities ≤ 2.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.