Description

6-Oxabicyclo[3.1.0]Hexan-2-Ol,4-(4-Morpholinyl)-,(1-α-,2-α-,4-α-,5-α-)-(9Ci) is a high-purity, advanced pharmaceutical intermediate featuring a complex oxabicyclo[3.1.0]hexane scaffold integrated with a morpholine moiety. This compound is valued for its unique stereochemistry and structural complexity, which are critical for imparting specific biological activity and selectivity in final drug molecules. It is primarily sought by research and development teams in the pharmaceutical and agrochemical industries for the synthesis of novel active ingredients.

Application

• Pharmaceutical Intermediate: A key chiral building block for the synthesis of novel therapeutic agents, particularly in central nervous system (CNS) and anti-infective drug discovery programs.
• Agrochemical Research: Used in the development of new-generation pesticides and herbicides, where its bicyclic structure can contribute to unique modes of action.
• Chemical Synthesis: Serves as a versatile precursor for further chemical elaboration in academic and industrial organic chemistry research.
• Ligand & Catalyst Development: The morpholine and constrained bicyclic structure make it a candidate for developing novel chiral ligands or organocatalysts for asymmetric synthesis.

Basic Information

Product Name	6-Oxabicyclo[3.1.0]Hexan-2-Ol,4-(4-Morpholinyl)-,(1-α-,2-α-,4-α-,5-α-)-(9Ci)
CAS No.	84845-80-7
Molecular Formula	C9H15NO3
Molecular Weight	185.22 g/mol
Synonyms	4-(Morpholin-4-yl)-6-oxabicyclo[3.1.0]hexan-2-ol; (1α,2α,4α,5α)-4-Morpholino-6-oxabicyclo[3.1.0]hexan-2-ol; 6-Oxabicyclo[3.1.0]hexan-2-ol, 4-(4-morpholinyl)-, (1α,2α,4α,5α)-; 84845-80-7; 4-Morpholino-6-oxabicyclo[3.1.0]hexan-2-ol (stereoisomer)
EINECS	Contact for details

Quality Control

Every batch of this advanced intermediate is produced under strict quality management systems. We employ state-of-the-art analytical techniques including HPLC, GC, and NMR to ensure identity, purity, and stereochemical integrity. A comprehensive Certificate of Analysis (COA) detailing purity, chiral purity, and residual solvent levels is provided with each shipment to support your regulatory and R&D documentation needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (typically 15-25°C). Keep away from incompatible materials. For long-term storage, consider storing under an inert atmosphere to maintain optimal stability.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Chiral Purity (Chiral HPLC)	≥ 98.0% ee
Water Content (KF)	≤ 0.5%
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.