Description

2,6-Dimethoxy-4-([(Pyridin-3-Ylmethyl)-Amino]-Methyl)-Phenol is a high-purity synthetic organic compound featuring a phenolic core substituted with dimethoxy and aminomethylpyridine groups. This unique molecular structure makes it a valuable advanced pharmaceutical intermediate and a versatile building block for medicinal chemistry research. It is primarily utilized by R&D chemists and process development scientists in the pharmaceutical and fine chemical industries for the synthesis of novel active pharmaceutical ingredients (APIs) and other complex molecules.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of novel drug candidates, particularly in central nervous system (CNS) and anti-infective research.
• Medicinal Chemistry Research: Used as a scaffold or precursor for structure-activity relationship (SAR) studies and lead optimization in drug discovery programs.
• Ligand Synthesis: Serves as a precursor for creating complex ligands used in catalysis and metal-organic frameworks (MOFs).
• Fine Chemical Synthesis: Employed in the multi-step synthesis of specialty chemicals, agrochemicals, and other high-value organic compounds.
• Bioconjugation Chemistry: The phenolic and amine functional groups allow for potential use in developing linkers for antibody-drug conjugates (ADCs) or other bioconjugates.

Basic Information

Product Name	2,6-Dimethoxy-4-([(Pyridin-3-Ylmethyl)-Amino]-Methyl)-Phenol
CAS No.	680185-77-7
Molecular Formula	C₁₅H₁₈N₂O₃
Molecular Weight	274.32 g/mol
Synonyms	4-[(Pyridin-3-ylmethyl)amino]methyl-2,6-dimethoxyphenol; 2,6-Dimethoxy-4-{[(pyridin-3-ylmethyl)amino]methyl}phenol; Phenol, 2,6-dimethoxy-4-[[(3-pyridinylmethyl)amino]methyl]-; 3-{[(3,5-Dimethoxy-4-hydroxyphenyl)methyl]amino}methylpyridine; 680185-77-7
EINECS	Contact for details

Quality Control

Our 2,6-Dimethoxy-4-([(Pyridin-3-Ylmethyl)-Amino]-Methyl)-Phenol is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC for purity and identity confirmation (IR, NMR), to ensure it meets the high standards required for pharmaceutical R&D and fine chemical synthesis. A comprehensive Certificate of Analysis (COA) detailing all specifications is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at controlled room temperature (15-25°C) under an inert atmosphere (e.g., nitrogen or argon) to prevent oxidation. Keep away from heat and incompatible materials.

Specification

Item	Specification
Appearance	White to off-white powder
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.