Description

tert-Butyl [(1R,2S,5S)-2-Amino-5-[(Dimethylamino)Carbonyl]Cyclohexyl]Carbamate Oxalate is a high-purity, chiral intermediate of significant importance in advanced pharmaceutical synthesis. Its value lies in its defined stereochemistry and protected functional groups, which are critical for constructing complex, biologically active molecules. This compound is primarily needed by research institutions and pharmaceutical companies engaged in the development of novel therapeutics, particularly for creating peptidomimetics and other targeted drug candidates.

Application

• Pharmaceutical Intermediate: A key chiral building block in the synthesis of complex active pharmaceutical ingredients (APIs).
• Peptidomimetic Research: Used to construct non-peptide scaffolds that mimic the structure and function of natural peptides for drug discovery.
• Protease Inhibitor Development: Serves as a core structure in the research and development of enzyme inhibitors.
• Chemical Biology & Medicinal Chemistry: Employed in structure-activity relationship (SAR) studies and lead optimization processes.
• Asymmetric Synthesis: Utilized in stereoselective reactions to introduce specific chiral centers into target molecules.
• Custom Synthesis & Contract Manufacturing: Supplied for custom synthesis projects requiring high-fidelity chiral intermediates.

Basic Information

Product Name	tert-Butyl [(1R,2S,5S)-2-Amino-5-[(Dimethylamino)Carbonyl]Cyclohexyl]Carbamate Oxalate
CAS No.	1210348-34-7
Molecular Formula	C16H29N3O6 • C2H2O4
Molecular Weight	Contact for details
Synonyms	(1R,2S,5S)-2-[(tert-Butoxycarbonyl)amino]-5-(dimethylcarbamoyl)cyclohexanaminium oxalate; Boc-Dap(Dimethylamide)-OH•Oxalate; tert-Butyl N-[(1R,2S,5S)-2-amino-5-(dimethylcarbamoyl)cyclohexyl]carbamate oxalate; (1R,2S,5S)-2-Amino-5-(dimethylcarbamoyl)cyclohexylcarbamic acid tert-butyl ester oxalate; Boc-Dap(NMe2)-OH oxalate salt; Chiral cyclohexane derivative oxalate salt
EINECS	Contact for details

Quality Control

Our tert-Butyl [(1R,2S,5S)-2-Amino-5-[(Dimethylamino)Carbonyl]Cyclohexyl]Carbamate Oxalate is manufactured under strict quality management systems to ensure batch-to-batch consistency and high purity suitable for research and development. Each lot undergoes rigorous analytical testing, including chiral purity verification and impurity profiling. Certificates of Analysis (COA) detailing identity, assay, chiral purity, and related substances are available upon request to support your regulatory and quality assurance needs.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled under dry conditions to maintain stability and purity.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Chiral Purity (Chiral HPLC)	≥ 99.0% ee
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm
Related Substances (HPLC)	Total impurities ≤ 2.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.