Description

3-[(Methylamino)Methyl]Azetidine, 3-Boc Protected Hydrochloride is a high-purity, protected amine building block essential for advanced organic synthesis. This compound is a critical intermediate in the development of novel active pharmaceutical ingredients (APIs) and fine chemicals, offering a versatile scaffold for medicinal chemistry. It is primarily utilized by research institutions and pharmaceutical companies engaged in drug discovery and process development.

Application

• Pharmaceutical Intermediate: A key building block in the synthesis of complex drug candidates, particularly in medicinal chemistry programs.
• Protease Inhibitor Research: Used in the development of novel protease inhibitors for therapeutic applications.
• Peptidomimetic Synthesis: Serves as a constrained scaffold for creating peptidomimetics with enhanced metabolic stability.
• Ligand and Catalyst Development: Employed in the preparation of specialized ligands and organocatalysts for asymmetric synthesis.
• Chemical Biology Probes: Useful for constructing molecular probes to study biological pathways and protein function.
• Custom Synthesis: A starting material for contract research and manufacturing organizations (CROs/CMOs) producing bespoke compounds.

Basic Information

Product Name	3-[(Methylamino)Methyl]Azetidine, 3-Boc Protected Hydrochloride
CAS No.	1170019-97-2
Molecular Formula	C11H23ClN2O2
Molecular Weight	250.77 g/mol
Synonyms	1-Boc-3-[(Methylamino)Methyl]Azetidine Hydrochloride; tert-Butyl 3-[(Methylamino)Methyl]Azetidine-1-carboxylate Hydrochloride; 3-(Methylaminomethyl)azetidine-1-carboxylic Acid tert-Butyl Ester Hydrochloride; 1-(tert-Butoxycarbonyl)-3-[(methylamino)methyl]azetidine Hydrochloride; 3-Boc-3-azetidinemethylamine, N-Methyl Hydrochloride; Azetidine, 3-[(methylamino)methyl]-, 1-(1,1-dimethylethyl) ester, hydrochloride (1:1); 3-(N-Methylaminomethyl)-1-Boc-azetidine HCl
EINECS	Contact for details

Quality Control

Our 3-[(Methylamino)Methyl]Azetidine, 3-Boc Protected Hydrochloride is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing, including HPLC, NMR, and mass spectrometry, to ensure identity, purity, and consistency. Certificates of Analysis (COA) with full traceability are provided and available upon request.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated area at a controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and should be handled under anhydrous conditions to maintain stability.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Identification (NMR)	Conforms to structure
Purity (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.