Tinib Antineoplastic Drugs

Tinib Antineoplastic Drugs

Tinib antineoplastic drugs are a major class of targeted cancer therapies that inhibit dysregulated tyrosine kinases or serine/threonine kinases involved in tumor growth, angiogenesis, and metastasis. Represented by imatinib, erlotinib, gefitinib, sunitinib, sorafenib, and numerous next-generation inhibitors, these APIs block oncogenic signaling pathways such as EGFR, VEGFR, PDGFR, BCR-ABL, ALK, and RET. Their precision targeting enables high efficacy with reduced systemic toxicity compared to traditional chemotherapy. Tinib drugs are widely used in leukemia, lung cancer, renal cancer, gastrointestinal stromal tumors, and melanoma. Resistance caused by kinase mutations has led to the development of multi-targeted and mutation-specific inhibitors, making tinibs a cornerstone of precision oncology.

Regorafenib (Hydrochloride) CAS NO 835621-07-3

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CAS No.:835621-07-3

Grade:Pharmacy Grade

Content:99.90%

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Regorafenib CAS NO 835621-08-4

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CAS No.:835621-08-4

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Content:99.90%

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n-(3-Cyano-10-Methyl-5-Oxo-1-Pentyl-1,5-Dihydro-2H-Dipyrido[1,2-A:2,3-D]Pyrimidin-2-Ylidene)Benzamide CAS NO 844851-48-5

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CAS No.:844851-48-5

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Content:99.90%

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1,2-Dihydro-n-[4-Methoxy-3-(4-Methyl-1-Piperazinyl)Phenyl]-3H-Benz[E]Indole-3-Carboxamide Hydrochloride CAS NO 847871-78-7

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CAS No.:847871-78-7

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4-Defluoro-4-Hydroxy Gefitinib CAS NO 847949-50-2

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CAS No.:847949-50-2

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Sphinx CAS NO 848057-98-7

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CAS No.:848057-98-7

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Fgfr Inhibitor CAS NO 848318-25-2

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CAS No.:848318-25-2

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