Description

4-(Bromoacetamido)Benzyl-1-Iodocarazolol is a specialized, high-purity biochemical building block designed for advanced research and development. This compound is of significant value for its role as a key intermediate in the synthesis of novel, high-affinity ligands and probes targeting adrenergic receptors. It is primarily needed by pharmaceutical R&D teams, academic research institutions, and biotechnology companies engaged in molecular pharmacology, radiopharmaceutical development, and receptor characterization studies.

Application

• Pharmaceutical Research: Critical intermediate in the synthesis of novel β-adrenergic receptor (β-AR) antagonists and imaging agents.
• Bioconjugation & Probe Development: The bromoacetamido moiety enables site-specific conjugation to proteins, peptides, or other biomolecules for creating targeted molecular probes.
• Receptor Binding Studies: Used to develop radiolabeled (e.g., with I-125 or I-131) or fluorescent derivatives for in vitro and in vivo receptor mapping and occupancy assays.
• Medicinal Chemistry: Serves as a versatile scaffold for structure-activity relationship (SAR) studies to optimize drug candidates targeting G-protein coupled receptors (GPCRs).
• Diagnostic Agent Precursor: A key starting material for developing potential PET (Positron Emission Tomography) or SPECT (Single-Photon Emission Computed Tomography) tracers for cardiac or neurological imaging.

Basic Information

Product Name	4-(Bromoacetamido)Benzyl-1-Iodocarazolol
CAS No.	97458-57-6
Molecular Formula	Contact for details
Molecular Weight	Contact for details
Synonyms	4-(Bromoacetamido)benzyl 1-iodocarazolol; 1-Iodocarazolol, 4-(bromoacetamido)benzyl ester; Carazolol derivative, iodinated; β-Adrenergic receptor ligand intermediate; BRL-4-(BrAc)benzyl-1-Iodo; (RS)-1-(4-(Bromoacetamido)benzyl)-4-(3-iodo-9H-carbazol-9-yl)butan-2-ol (tentative structure-based name)
EINECS	Contact for details

Quality Control

Our 4-(Bromoacetamido)Benzyl-1-Iodocarazolol is produced under strict quality management protocols to ensure batch-to-batch consistency and high purity, essential for sensitive research applications. Each lot undergoes comprehensive analytical characterization, including HPLC for purity and identity confirmation via spectroscopic methods. A Certificate of Analysis (COA) detailing all specifications is provided with every shipment.

Storage

Preserve in a tightly closed container, protected from light. Store in a freezer at -20°C or below under inert atmosphere for long-term stability. Allow the sealed container to reach room temperature before opening to minimize moisture condensation. Keep away from strong oxidizing agents.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (HPLC)	Conforms to reference standard
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 95% (Area %)
Water Content (KF)	≤ 1.0 %
Residual Solvents (GC)	Meets ICH guidelines

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.