Description

1-Benzyl-3-Methanesulfonyloxyazetidine is a high-purity, functionalized azetidine derivative of significant interest in advanced organic synthesis. This compound serves as a versatile and critical building block, particularly valued for its reactive mesylate leaving group, which facilitates nucleophilic substitution reactions. It is primarily sought after by research institutions and pharmaceutical companies engaged in the development of novel active pharmaceutical ingredients (APIs) and other fine chemicals, where precise molecular construction is paramount.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of complex drug candidates, especially those containing the azetidine pharmacophore.
• Organic Synthesis Building Block: Used in nucleophilic substitution reactions to introduce the benzyl-protected azetidine moiety into larger molecular frameworks.
• Agrochemical Research: Employed in the development of new crop protection agents and herbicides.
• Material Science: Potential monomer or modifier in the creation of specialized polymers with unique properties.
• Chemical Biology Probes: Useful for labeling or modifying biomolecules in research settings to study biological pathways.

Basic Information

Product Name	1-Benzyl-3-Methanesulfonyloxyazetidine
CAS No.	67160-49-0
Molecular Formula	C11H15NO3S
Molecular Weight	241.31 g/mol
Synonyms	3-(Methylsulfonyloxy)-1-benzylazetidine; 1-Benzylazetidin-3-yl methanesulfonate; Azetidine, 1-benzyl-3-[(methylsulfonyl)oxy]-; 1-Benzyl-3-(methylsulfonyloxy)azetidine; 1-Benzyl-3-mesyloxyazetidine; 3-Methanesulfonyloxy-1-benzylazetidine
EINECS	Contact for details

Quality Control

Our 1-Benzyl-3-Methanesulfonyloxyazetidine is manufactured under strict quality control protocols to ensure batch-to-batch consistency and high purity suitable for research and development applications. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing key parameters such as purity (by HPLC/NMR), identity confirmation, and impurity profiles. Our quality management system is designed to meet the stringent requirements of our global B2B clientele.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). This product is hygroscopic (moisture-sensitive) and should be handled under anhydrous conditions to maintain stability and purity.

Specification

Item	Specification
Appearance	White to off-white solid
Identification (IR)	Conforms to structure
Purity (HPLC)	≥ 97.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.