Description

5-(Aminosulfonyl)-2-Morpholin-4-Ylbenzoic Acid is a high-purity, multifunctional organic building block characterized by its benzoic acid core substituted with a sulfonamide and a morpholine group. This compound matters for its role as a critical intermediate in the synthesis of complex molecules, particularly in pharmaceutical research and development. It is primarily needed by R&D chemists and process development scientists in the pharmaceutical, agrochemical, and specialty chemical industries for creating novel active ingredients and functional materials.

Application

• Pharmaceutical Intermediate: A key synthon in the research and production of potential drug candidates, particularly those targeting enzymes or receptors where the sulfonamide and morpholine pharmacophores are relevant.
• Agrochemical Synthesis: Used in the development of new herbicides, fungicides, or plant growth regulators that incorporate its specific aromatic substitution pattern.
• Chemical Research & Development: Serves as a versatile building block for constructing more complex heterocyclic compounds and functionalized aromatic systems in academic and industrial labs.
• Material Science Precursor: Potential use in the synthesis of specialty polymers, ligands for catalysis, or organic electronic materials due to its multifunctional nature.
• Bioconjugation & Probe Development: The carboxylic acid and sulfonamide groups offer handles for conjugation, making it useful for creating biochemical probes or labeled compounds.

Basic Information

Item	Details
Product Name	5-(Aminosulfonyl)-2-Morpholin-4-Ylbenzoic Acid
CAS No.	65194-68-5
Molecular Formula	C11H14N2O5S
Molecular Weight	286.31 g/mol
Synonyms	2-Morpholino-5-sulfamoylbenzoic acid; 5-Sulfamoyl-2-morpholinobenzoic acid; Benzoic acid, 5-(aminosulfonyl)-2-morpholino-; 5-Carboxy-2-morpholinobenzenesulfonamide; 65194-68-5; 2-Morpholin-4-yl-5-sulfamoylbenzoic acid
EINECS	Contact for details

Quality Control

Our 5-(Aminosulfonyl)-2-Morpholin-4-Ylbenzoic Acid is manufactured under strict quality management systems. Each batch undergoes rigorous analytical testing to ensure identity, purity, and consistency. We provide comprehensive Certificates of Analysis (COA) with each shipment, detailing key parameters such as assay, impurity profile, and physical characteristics. Our quality commitment aligns with cGMP principles where applicable, supporting its use in regulated research and development.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed after opening to prevent degradation from atmospheric moisture. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Loss on Drying	≤ 1.0%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 20 ppm
Related Substances (HPLC)	Total impurities ≤ 2.0% Any single impurity ≤ 0.5%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.