Description

4-Iodo-n-(2-Morpholin-4-Yl-Ethyl)-Benzenesulfonamide is a specialized sulfonamide derivative featuring a morpholinoethyl side chain and an iodine substituent, making it a valuable synthetic intermediate. This compound is engineered for high-purity applications where precise molecular architecture is critical for downstream performance. It is primarily targeted at research and development chemists in the pharmaceutical and agrochemical industries for use in medicinal chemistry, particularly in the synthesis of targeted bioactive molecules and as a key building block in drug discovery programs.

Application

• Pharmaceutical Intermediate: Serves as a crucial building block in the synthesis of novel drug candidates, especially those targeting enzyme inhibition or receptor modulation.
• Medicinal Chemistry Research: Used in structure-activity relationship (SAR) studies and lead optimization due to its unique sulfonamide and halogenated aromatic structure.
• Agrochemical Development: Acts as a precursor in the creation of new herbicides or fungicides where the iodine atom and sulfonamide group confer specific biological activity.
• Chemical Biology Probes: Utilized in the development of molecular probes and labeled compounds for biochemical and diagnostic research.
• Organic Synthesis: Functions as a versatile intermediate for cross-coupling reactions (e.g., Suzuki, Sonogashira) and further functionalization of the aromatic ring.
• Library Synthesis: Employed in combinatorial chemistry for generating diverse compound libraries for high-throughput screening.

Basic Information

Product Name	4-Iodo-n-(2-Morpholin-4-Yl-Ethyl)-Benzenesulfonamide
CAS No.	433688-20-1
Molecular Formula	C12H17IN2O3S
Molecular Weight	396.25 g/mol
Synonyms	4-Iodo-N-(2-morpholinoethyl)benzenesulfonamide; Benzenesulfonamide, 4-iodo-N-(2-(4-morpholinyl)ethyl)-; N-(2-Morpholin-4-ylethyl)-4-iodobenzenesulfonamide; 4-Iodo-N-(2-(morpholin-4-yl)ethyl)benzenesulfonamide; 433688-20-1; 4-Iodo-N-(2-morpholin-4-ylethyl)benzenesulfonamide
EINECS	Contact for details

Quality Control

Our 4-Iodo-n-(2-Morpholin-4-Yl-Ethyl)-Benzenesulfonamide is manufactured under strict quality control protocols to ensure batch-to-batch consistency and high purity suitable for research and development. Each lot is accompanied by a comprehensive Certificate of Analysis (COA) detailing purity, identity, and impurity profiles. We adhere to cGMP principles where applicable, and our quality systems are designed to meet the stringent requirements of pharmaceutical and fine chemical industries.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry, and well-ventilated place at a controlled room temperature (15-25°C). Due to its hygroscopic (moisture-sensitive) nature, the container must be kept tightly sealed after opening to prevent degradation from atmospheric moisture. Keep away from incompatible materials.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Water Content (KF)	≤ 0.5%
Residue on Ignition	≤ 0.1%
Heavy Metals	≤ 10 ppm
Single Unknown Impurity (HPLC)	≤ 0.5%
Total Impurities (HPLC)	≤ 2.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.