Description

Ethyl 5-[[Amino(Imino)Methyl]Amino]-2-(Benzoylamino)Pentanoate Hydrochloride is a high-purity, non-natural amino acid derivative of significant interest in advanced organic synthesis. This compound serves as a critical building block for the development of novel bioactive molecules, particularly those targeting specific enzymatic pathways. It is primarily utilized by pharmaceutical research and development organizations, as well as by fine chemical manufacturers specializing in custom peptide mimetics and enzyme inhibitors.

Application

• Pharmaceutical Intermediate: A key precursor in the synthesis of novel drug candidates, particularly protease inhibitors and other enzyme-targeted therapeutics.
• Peptidomimetic Research: Used to construct modified peptide backbones that mimic natural peptides but with enhanced metabolic stability and bioavailability.
• Bioconjugation Chemistry: Serves as a linker or functional handle for attaching payloads in antibody-drug conjugate (ADC) and prodrug development.
• Chemical Biology Probes: Employed in the design and synthesis of activity-based probes (ABPs) for studying enzyme function and mechanism.
• Agrochemical Research: Investigated as a component in the development of new crop protection agents with specific biological activity.
• Academic & Institutional R&D: Used in university and research institute laboratories for fundamental studies in medicinal chemistry and biochemistry.

Basic Information

Item	Detail
Product Name	Ethyl 5-[[Amino(Imino)Methyl]Amino]-2-(Benzoylamino)Pentanoate Hydrochloride
CAS No.	128805-94-7
Molecular Formula	C15H23N5O3 • HCl
Molecular Weight	373.84 g/mol (Free base: 321.38 g/mol)
Synonyms	Ethyl 5-(amidinoamino)-2-(benzamido)pentanoate hydrochloride; Ethyl 5-guanidino-2-benzamidopentanoate hydrochloride; 2-Benzamido-5-guanidinopentanoic acid ethyl ester hydrochloride; N2-Benzoyl-N5-(diaminomethylene)-L-ornithine ethyl ester hydrochloride; L-Ornithine, N2-benzoyl-N5-(diaminomethylene)-, ethyl ester, hydrochloride; AG-1478 derivative; Tyrphostin AG 1478 analog
EINECS	Contact for details

Quality Control

Our Ethyl 5-[[Amino(Imino)Methyl]Amino]-2-(Benzoylamino)Pentanoate Hydrochloride is manufactured under a strict quality management system. Each batch undergoes comprehensive analytical testing to ensure identity, purity, and consistency. We provide a detailed Certificate of Analysis (COA) with every shipment, which includes data from HPLC, NMR, and mass spectrometry. Our quality commitment aligns with the standards expected for pharmaceutical-grade intermediates in global supply chains.

Storage

Preserve in a tightly closed container, protected from light. Store in a cool, dry place at a controlled room temperature (15-25°C). This compound is hygroscopic (moisture-sensitive) and should be handled in a dry environment to prevent degradation. For long-term storage, consider desiccant or inert atmosphere conditions.

Specification

Item	Specification
Appearance	White to off-white crystalline powder
Identification (HPLC)	Conforms to reference standard
Identification (IR)	Conforms to structure
Assay (HPLC)	≥ 98.0%
Water Content (KF)	≤ 1.0%
Residue on Ignition	≤ 0.5%
Heavy Metals	≤ 20 ppm
Related Substances (HPLC)	Total impurities ≤ 2.0%

Note: Specifications can be tailored. Please contact us for the detailed technical data sheet of a specific grade.